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3D structures from the PDB for "Tyrosine-protein kinase ABL1 [201-500,E255K]" AND "BDBM13530"
(Proteins have >= 85% sequence identity and ligands are exact matches)


Seq IdentityJmol DisplayPDB Title
2HYY>99%JmolHUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC)
6NPE>99%JmolC-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD6), 2-CYANO-N-(4-(3,4- DICHLOROPHENYL)THIAZOL-2-YL)ACETAMIDE
6NPV>99%JmolC-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD51), N-(1-(3,4- DICHLOROPHENYL)-4-(2-HYDROXYETHYL)-4,5-DIHYDRO-1H-PYRAZOL-3-YL) ISONICOTINAMIDE
6NPU>99%JmolC-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD29), N-(1-(3,4- DICHLOROPHENYL)-4,5-DIHYDRO-1H-PYRAZOL-3-YL)ACETAMIDE
3PYY>99%JmolDISCOVERY AND CHARACTERIZATION OF A CELL-PERMEABLE, SMALL-MOLECULE C- ABL KINASE ACTIVATOR THAT BINDS TO THE MYRISTOYL BINDING SITE
7N9G>99%JmolCRYSTAL STRUCTURE OF THE ABL 1B KINASE DOMAIN IN COMPLEX WITH DASATINIB AND IMATINIB
3MS9>99%JmolABL KINASE IN COMPLEX WITH IMATINIB AND A FRAGMENT (FRAG1) IN THE MYRISTATE POCKET
6HD4>99%JmolABL1 IN COMPLEX WITH COMPOUND 7 AND IMATINIB (STI-571)
6HD6>99%JmolABL1 IN COMPLEX WITH COMPOUND6 AND IMATINIB (STI-571)
1IEP>99%JmolCRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571.
1OPJ>99%JmolSTRUCTURAL BASIS FOR THE AUTO-INHIBITION OF C-ABL TYROSINE KINASE